Hhdpharm Supply Regorafenib Anticancer Inhibitor Raw Material Regorafenib Powder CAS 755037-03-7

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Wuhan Hengheda Pharm Co., Ltd.

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Product Description

Wuhan HHD Supply Regorafenib Anticancer Inhibitor Raw Material Regorafenib Powder CAS 755037-03-7 
 

Basic information:

 
Prodcut nameRegorafenib
Synonyms 4-(4-(3-(4-Chloro-3-(trifluoromethyl)phenyl)ureido)-3-fluorophenoxy)-N-methylpicolinamide;4-[4-({[4-Chloro-3-(trifluoromethyl)phenyl]carbamoyl}amino)-3-fluorophenoxy]-N-methylpyridine-2-carboxamide;Stivarga®;4-[4-[[4-chloro-3-(trifluoromethyl)phenyl]carbamoylamino]-3-fluorophenoxy]-N-methylpyridine-2-carboxamide;
MOQ10g
CAS755037-03-7
AppearancePowder
Molecular FormulaC21H15ClF4N4O3
Molecular Weight482.815
Assay99%
ApplicationPharma grade
PackingAs per your request
StoragePreserve in tight, light-resistant containers in a cool place

Description:

Regorafenib (BAY 73-4506, commercial name Stivarga) is an oral multi-kinase inhibitor developed by Bayer which targets angiogenic, stromal and oncogenic receptor tyrosine kinase (RTK). Regorafenib shows anti-angiogenic activity due to its dual targeted VEGFR2-TIE2 tyrosine kinase inhibition. Since 2009 it was studied as a potential treatment option in multiple tumor types.[1] By 2015 it had 2 US approvals for advanced cancers.

 

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